S
Santos Fustero
Researcher at University of Valencia
Publications - 370
Citations - 10515
Santos Fustero is an academic researcher from University of Valencia. The author has contributed to research in topics: Enantioselective synthesis & Catalysis. The author has an hindex of 39, co-authored 365 publications receiving 8865 citations. Previous affiliations of Santos Fustero include University of Barcelona & Janssen Pharmaceutica.
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Fluorine in pharmaceutical industry: fluorine-containing drugs introduced to the market in the last decade (2001-2011).
Jiang Wang,María Sánchez-Roselló,José Luis Aceña,Carlos del Pozo,Alexander E. Sorochinsky,Alexander E. Sorochinsky,Alexander E. Sorochinsky,Santos Fustero,Vadim A. Soloshonok,Vadim A. Soloshonok,Hong Liu +10 more
TL;DR: Introduced to the Market in the Last Decade (2001−2011) Jiang Wang,† María Sańchez-Rosello,́‡,§ Jose ́ Luis Aceña, Carlos del Pozo,‡ and Hong Liu.
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From 2000 to mid-2010: a fruitful decade for the synthesis of pyrazoles.
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Fluorine-Containing Drugs Approved by the FDA in 2018
Haibo Mei,Jianlin Han,Santos Fustero,Mercedes Medio-Simón,Daniel M. Sedgwick,Claudio Santi,Renzo Ruzziconi,Vadim A. Soloshonok,Vadim A. Soloshonok +8 more
TL;DR: The newly approved pharmaceuticals feature several types of aromatic F- and CF3-, aliphatic (CF2) substitution, offering advances in treatment of various diseases, including cancer, HIV, malarial and smallpox infections.
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Recent Advances in the Synthesis of Pyrazoles. A Review
TL;DR: A five-membered, two-nitrogen-containing heterocycle ring is widely found as the core structure in a large variety of compounds that possess important agrochemical and pharmacological properties as mentioned in this paper.
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Improved regioselectivity in pyrazole formation through the use of fluorinated alcohols as solvents: synthesis and biological activity of fluorinated tebufenpyrad analogs.
Santos Fustero,Raquel Román,Juan F. Sanz-Cervera,Antonio Simón-Fuentes,Ana C. Cuñat,Salvador Villanova,Marcelo Murguia +6 more
TL;DR: The use of fluorinated alcohols such as 2,2,2-trifluoroethanol (TFE) and 1,1,3,3-hexafluoro-2-propanol (HFIP) as solvents dramatically increases the regioselectivity in the pyrazole formation, and this modification is used in a straightforward synthesis of fluorination analogs of Tebufenpyrad with acaricide activity.