M
Marco Santagostino
Researcher at Boehringer Ingelheim
Publications - 75
Citations - 912
Marco Santagostino is an academic researcher from Boehringer Ingelheim. The author has contributed to research in topics: Catalysis & Aryl. The author has an hindex of 15, co-authored 72 publications receiving 890 citations. Previous affiliations of Marco Santagostino include Sigma-Tau & University of Milan.
Papers
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Journal ArticleDOI
Oxidation of Alcohols with o-Iodoxybenzoic Acid in DMSO: A New Insight into an Old Hypervalent Iodine Reagent
Patent
Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions
Stephan Georg Mueller,Klaus Rudolf,Philipp Lustenberger,Dirk Stenkamp,Alexander Dreyer,Kirsten Arndt,Gerhard Schaenzle,Henri Doods,Marco Santagostino,Fabio Paleari +9 more
TL;DR: In this article, the CGRP antagonists of general formula A and R 1 to R 3 are defined as tautomers, diastereomers, enantiomers, hydrates thereof, the mixtures thereof and the salts thereof, particularly the physiologically acceptable salts thereof with inorganic or organic acids.
Patent
CCR2 receptor antagonists and uses thereof
Heiner Ebel,Sara Frattini,Kai Gerlach,Riccardo Giovannini,Christoph Hoenke,Rocco Mazzaferro,Marco Santagostino,Stefan Scheuerer,Christofer S. Tautermann,Thomas Trieselmann +9 more
TL;DR: In this article, novel antagonists for CCR2 (CC chemokine receptor 2) and their use for providing medicaments for treating conditions and diseases, especially pulmonary diseases like asthma and COPD.
Journal ArticleDOI
2‐(Tributylstannyl)‐1‐{[2‐(trimethylsilyl)ethoxy]methyl}‐1H‐indole: Synthesis and use as a 1H‐indol‐2‐yl‐anion equivalent
TL;DR: Pd-catalyzed reaction of 2-(tributylstannyl)-1-{[2-(trimethylsilyl)ethoxy]methyl}-1H-indole (5) with a variety of aryl, hetero-aryl, vinyl, and allyl halides provides an efficient entry to the corresponding cross-coupled products as mentioned in this paper.
Patent
Selected cgrp antagonists, methods for the production thereof and their use as medicaments
Stephan Georg Mueller,Klaus Rudolf,Philipp Lustenberger,Dirk Stenkamp,Alexander Dreyer,Kirsten Arndt,Henri Doods,Gerhard Schaenzle,Marco Santagostino,Fabio Paleari +9 more
TL;DR: In this article, the CGRP antagonists of general formula (I) are defined as in Claim 1, to their tautomers, isomers, diastereomers, enantiomers, hydrates, mixtures and their salts as well as the hydrate of the salts, particularly their physiologically compatible salts having inorganic or organic acids.