Showing papers by "Valérie Collot published in 2005"
TL;DR: Three 5-bromo-3-iodoindoles and two indazoles have been studied with respect to their reactivity and selectivity in palladium catalyzed Sonogashira and Suzuki cross-coupling reactions to obtain a large range of new functionalized indoles and indazole ligands, which are potential 5-HT receptor ligands.
Abstract: 3-Iodoindoles, 5-bromo-3-iodoindoles and 5-bromo-3-iodoindazoles have been studied with respect to their reactivity and selectivity in palladium catalyzed Sonogashira and Suzuki cross-coupling reactions. As a result, sequential Sonogashira-Sonogashira, Sonogashira-Suzuki, and Suzuki-Sonogashira reactions with 5-bromo-3-iodoindoles or indazoles were used to obtain a large range of new functionalized indoles and indazoles, which are potential 5-HT receptor ligands.
39 citations
TL;DR: In this article, the reactivity and selectivity of 5.3-Iodoindoles, 5.bromo-3-iodoindoles and 5.5-bromodioxindoles have been studied with respect to their reactivity in palladium catalyzed Sonogashira and Suzuki cross-coupling reactions.
Abstract: 3-Iodoindoles, 5-bromo-3-iodoindoles and 5-bromo-3-iodoindazoles have been studied with respect to their reactivity and selectivity in palladium catalyzed Sonogashira and Suzuki cross-coupling reactions. As a result, sequential Sonogashira-Sonogashira, Sonogashira-Suzuki, and Suzuki-Sonogashira reactions with 5-bromo-3-iodoindoles or indazoles were used to obtain a large range of new functionalized indoles and indazoles, which are potential 5-HT receptor ligands.
1 citations