S
Shinichiro Fuse
Researcher at Nagoya University
Publications - 118
Citations - 1983
Shinichiro Fuse is an academic researcher from Nagoya University. The author has contributed to research in topics: Catalysis & Chemistry. The author has an hindex of 23, co-authored 108 publications receiving 1603 citations. Previous affiliations of Shinichiro Fuse include Harvard University & Tokyo Institute of Technology.
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Journal ArticleDOI
Efficient Amide Bond Formation through a Rapid and Strong Activation of Carboxylic Acids in a Microflow Reactor
TL;DR: The development of highly efficient amide bond forming methods which are devoid of side reactions, including epimerization, is important, and such a method is described herein and is based on the concept of rapid and strong activation of carboxylic acids.
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A formal total synthesis of taxol aided by an automated synthesizer.
Takayuki Doi,Shinichiro Fuse,Shigeru Miyamoto,Kazuoki Nakai,Daisuke Sasuga,Takashi Takahashi +5 more
TL;DR: A 36-step synthesis was carried out in automated synthesizers to provide a synthetic key intermediate of taxol using a microwave-assisted alkylation reaction to construct the ABC ring system from an AC precursor.
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Structural analysis of the contacts anchoring moenomycin to peptidoglycan glycosyltransferases and implications for antibiotic design
TL;DR: A novel moenomycin intermediate is prepared that maintains these six contacts but does not contain the putative minimal pharmacophore and may facilitate the design of antibiotics targeted against peptidoglycan glycosyltransferases.
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Recent progresses in the synthesis of functionalized isoxazoles
TL;DR: A comprehensive survey of the recent new synthetic approaches to functionalized isoxazoles, with particular focus on the last three years with regard to the following reaction types: (1) 1,3-dipolar cycloaddition, (2) condensation, (3) cycloisomerization, and (4) direct functionalization.
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Continuous-flow synthesis of vitamin D3
Shinichiro Fuse,Nobutake Tanabe,Masahito Yoshida,Hayato Yoshida,Takayuki Doi,Takashi Takahashi +5 more
TL;DR: A highly efficient, two-stage, continuous-flow synthesis of vitamin D(3) from provitamin D( 3) was achieved and required neither intermediate purification nor high-dilution conditions.