Journal ArticleDOI
N-Glycyl-β-glycopyranosylamines, Derivatives of Mono- and Disaccharides, and Their Use for the Preparation of Carboxylic Acid Glycoconjugates.
TLDR
In this article, a preparation procedure for the synthesis of N-glycyl-β-glycopyranosylamines, derivatives of monosaccharides (d-galactose,d-mannose,l-fucose, and N-acetyl-d-glucosamine) and disaccharide derivatives (lactoses, melibiose, cellobiose and maltose) was developed.Abstract:
A convenient preparative procedure was developed for the synthesis ofN-glycyl-β-glycopyranosylamines, derivatives of monosaccharides (d-galactose,d-mannose,l-fucose, andN-acetyl-d-glucosamine) and disaccharides (lactose, melibiose, cellobiose, and maltose). These compounds were demonstrated to be useful for the preparation of glycoconjugates of biologically active compounds containing the carboxy group (nicotinic, orotic, kynurenic, and indoleacetic acids). Synthetic pathways were developed for conversions ofN-glycyl-β-glycopyranosylamines into derivatives containing the carboxy group with the use of malonic andl-tartaric acid derivatives.read more
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Journal ArticleDOI
Synthesis of conjugates of polyhedral boron compounds with carbohydrates
A. V. Orlova,Leonid O. Kononov +1 more
TL;DR: In this article, the conjugates of polyhedral boron compounds with carbohydrates, potential third-generation agents for neutron capture therapy, are systematised and generalised.
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Journal ArticleDOI
N-glycyl-β-glycopyranosylamines, derivatives of mono- and disaccharides, and their use for the preparation of carboxylic acid glycoconjugates
TL;DR: In this article, a preparation procedure for the synthesis of N-glycyl-β-glycopyranosylamines, derivatives of monosaccharides (d-galactose,d-mannose,l-fucose, and N-acetyl-d-glucosamine) and disaccharide derivatives (lactoses, melibiose, cellobiose and maltose) was developed.