S
Stefano Moro
Researcher at University of Padua
Publications - 363
Citations - 12565
Stefano Moro is an academic researcher from University of Padua. The author has contributed to research in topics: Adenosine receptor & Receptor. The author has an hindex of 55, co-authored 329 publications receiving 10894 citations. Previous affiliations of Stefano Moro include Polaris Industries & University of North Carolina at Chapel Hill.
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Medicinal Chemistry and the Molecular Operating Environment (MOE): Application of QSAR and Molecular Docking to Drug Discovery
TL;DR: This work provides a brief description of a series of studies implemented in the software MOE (Molecular Operating Environment) with particular attention to the medicinal chemistry aspects.
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FAM/USP9x, a Deubiquitinating Enzyme Essential for TGFβ Signaling, Controls Smad4 Monoubiquitination
Sirio Dupont,Anant Mamidi,Michelangelo Cordenonsi,Marco Montagner,Luca Zacchigna,Maddalena Adorno,Graziano Martello,Michael J. Stinchfield,Sandra Soligo,Leonardo Morsut,Masafumi Inui,Stefano Moro,Nicola Modena,Francesco Argenton,Stuart J. Newfeld,Stefano Piccolo +15 more
TL;DR: This study defines a regulative ubiquitination step controlling Smads that is parallel to those impinging on R-Smad phosphorylation, and points to Smad4 monoubiquitinated and deubiquitination as a way for cells to set their TGFbeta responsiveness.
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The mitochondrial calcium uniporter is a multimer that can include a dominant-negative pore-forming subunit.
Anna Raffaello,Diego De Stefani,Davide Sabbadin,Enrico Teardo,Giulia Merli,Anne Picard,Vanessa Checchetto,Stefano Moro,Ildikò Szabò,Rosario Rizzuto +9 more
TL;DR: The structural complexity of MCU is unveiled and a novel regulatory mechanism, based on the inclusion of dominant‐negative subunits in a multimeric channel, that underlies the fine control of the physiologically and pathologically relevant process of mitochondrial calcium homeostasis is demonstrated.
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Bridging Molecular Docking to Molecular Dynamics in Exploring Ligand-Protein Recognition Process: An Overview.
Veronica Salmaso,Stefano Moro +1 more
TL;DR: An overview of the evolution of structure-based drug discovery techniques in the study of ligand-target recognition phenomenon, going from the static molecular docking toward enhanced molecular dynamics strategies is presented.
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Ciprofloxacin and levofloxacin attenuate microglia inflammatory response via TLR4/NF-kB pathway.
Morena Zusso,Valentina Lunardi,Davide Franceschini,Andrea Pagetta,Rita Lo,Stefano Stifani,Anna Chiara Frigo,Pietro Giusti,Stefano Moro +8 more
TL;DR: CPFX and LVFX inhibited LPS-induced secretion of pro-inflammatory cytokines and activation of NF-κB in primary microglia and might facilitate the development of new molecules directed at the TLR4–MD-2 complex, a potential key target for controlling neuroinflammation.