Journal ArticleDOI
Thiolysis of oxazolines: A new, selective method for the direct conversion of peptide oxazolines into thiazolines
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TLDR
In this paper, a direct oxazoline→thiazoline conversion can be realized by thiolysis of oxazolines with H2S in methanol/triethylamine, followed by cyclodehydration with Burgess reagent.About:
This article is published in Tetrahedron Letters.The article was published on 1995-09-04. It has received 90 citations till now. The article focuses on the topics: Burgess reagent & Thiolysis.read more
Citations
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Solvent-free heterocyclic synthesis.
TL;DR: 1. Six-Membered Heterocycles with One Heteroatom 4155 7.6.1.
Journal ArticleDOI
Thioamides as useful synthons in the synthesis of heterocycles.
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Bioactive peptides and depsipeptides with anticancer potential: sources from marine animals.
TL;DR: The immense potential of marine animals as bioactive peptide sources, since they have been found as secondary metabolites from sponges, ascidians, tunicates, and mollusks, is demonstrated.
Journal ArticleDOI
Recent Progress of the Synthetic Studies of Biologically Active Marine Cyclic Peptides and Depsipeptides
Yasumasa Hamada,Takayuki Shioiri +1 more
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Overview of the chemistry of 2-thiazolines.
TL;DR: An overview of the chemistry of 2-thiazolines, including new methodologies for their preparation, and recent applications, such as their growing use in organic synthesis in the biological field and asymmetric catalysis as ligands.
References
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Journal ArticleDOI
The chemistry of 2-oxazolines (1985–present)
Thomas G. Gant,Albert I. Meyers +1 more
TL;DR: The use of chiral oxazolines as ligands in asymmetric catalysis has been extensively studied in the literature as mentioned in this paper, with a large number of important publications detailing oxazoline-related chemistry, suggesting that research in this area, as in synthetic organic chemistry in general, has yet to mature.
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Bis(oxazoline)copper(II) complexes as chiral catalysts for the enantioselective Diels-Alder reaction
TL;DR: In this paper, the utility of chiral Cu(1I) bis(oxazoline) complexes as Lewis acid catalysts for the Diels-Alder reactions of unsubstituted acrylimides was investigated.
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