scispace - formally typeset
F

Fernando Albericio

Researcher at University of KwaZulu-Natal

Publications -  1012
Citations -  29912

Fernando Albericio is an academic researcher from University of KwaZulu-Natal. The author has contributed to research in topics: Peptide synthesis & Solid-phase synthesis. The author has an hindex of 76, co-authored 965 publications receiving 26146 citations. Previous affiliations of Fernando Albericio include University of Barcelona & University of Chile.

Papers
More filters
Journal ArticleDOI

Exploring solid-phase approaches for the preparation of new β-lactams from amino acids

TL;DR: Two solid-phase approaches, involving the base-assisted intramolecularalkylation of N-chloroacetyl-Phe derivatives anchored to appropriatesolid supports, were investigated for the preparation of novel β-lactams.
Journal ArticleDOI

Further applications of classical amide coupling reagents: Microwave-assisted esterification on solid phase

TL;DR: The robustness of this method relies on the use of classical solid‐phase coupling reagents, heating by microwave irradiation, and a short time period, which results in high yields and the minimization of racemization.
Journal ArticleDOI

2,2,4,6,7‐Pentamethyl‐2,3‐dihydrobenzofuran‐5‐methyl (Pbfm) as an Alternative to the Trityl Group for the Side‐Chain Protection of Cysteine and Asparagine/Glutamine

TL;DR: The benzyl derivative of the PBF group, which is the most commonly used side-chain protecting group for Arg, has been proposed for the protection of the side chains of Cys, Asp, and Glu.
Journal ArticleDOI

Understanding Tetrahydropyranyl as a Protecting Group in Peptide Chemistry.

TL;DR: Tetrahydropyranyl is a useful moiety for the side‐chain protection of serine, threonine and cysteine and is suitable for the Fmoc/tBu solid‐phase peptide synthesis strategy.
Journal ArticleDOI

Semipermanent p-nitrobenzyloxycarbonyl (pNZ) protection of Orn and Lys side chains: prevention of undesired α-Fmoc removal and application to the synthesis of cyclic peptides

TL;DR: Semipermanent side-chain protection of Orn and Lys with p-nitrobenzyloxycarbonyl (pNZ) for Fmoc/tBu chemistry does not result in the unwanted removal of α-Fmoc that occurs when groups such as Alloc are used for the same application as discussed by the authors.