Journal ArticleDOI
A Simple One-Step Synthesis of Substituted Methyl 2-Benzoylamino-3-arylaminopropenoates, Intermediates in the Preparation of Substituted Arylaminoalanines
TLDR
In this paper, a simple one-step synthesis of substituted methyl 2-benzolamino-3-anilinopropenoates 8a-r from substituted anilines 7a r and methyl 2.benzoylamino3-dimethylamin-opropoenates 6 is described.Abstract:
A simple one-step synthesis of substituted methyl 2-benzolamino-3-anilinopropenoates 8a-r from substituted anilines 7a-r and methyl 2-benzoylamino-3-dimethylaminopropenoates 6 is described.
Eine einfache, einstufige Synthese substituierter 2-Benzoylamino-3-arylaminopropensauremethylester, Zwischenprodukte fur die Herstellung substituierter Arylaminoaniline.
Eine einfache, einstufige Synthese der substituierten 2-Benzoylamino-3-arylaminopropensauremethylester 8a-r aus den substituierten Anilin-Derivaten 7a-r und 2-Benzoylamino-3-dimethylaminopropensauremethylester 6 wird beschrieben.read more
Citations
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Journal ArticleDOI
Synthesis of heterocycles from alkyl 3-(dimethylamino)propenoates and related enaminones.
Branko Stanovnik,Jurij Svete +1 more
Journal ArticleDOI
Parallel solution-phase synthesis of (Z)-3-(arylamino)-2,3-dehydroalanine derivatives and solid-phase synthesis of fused pyrimidones.
TL;DR: N-Protected (Z)-3-(arylamino)-2,3-dehydroalanine esters 5 and 10 were prepared in one step from methyl (Z)2-acylamino-3-(dimethylamino)prop-2-enoates 3 and 9 and anilines 4 employing a parallel solution-phase synthetic approach.
Journal ArticleDOI
Methyl 2‐benzoylamino‐3‐dimethylaminopropenoate in the synthesis of heterocyclic systems. An attempt to prepare benzoylamino substituted azolo‐ and azinopyrimidines with a bridgehead nitrogen atom
TL;DR: Methyl 2-benzoylamino-3-dimethylaminopropenoate (2) was introduced as a new reagent for the preparartion of fused pyrimidinones 4 from heterocyclic α-amino compounds in acetic acid as mentioned in this paper.
Journal ArticleDOI
Methyl 2-benzoylamino-3-dimethylaminopropenoate in the synthesis of fused pyranones. The synthesis of derivatives of tetrahydro-2H-1-benzopyran-2-one, isomeric 2H-naphtho[1,2-b]pyran-2-one and 3H-naphtho[2,1-b]pyran-3-one, pyrano[3,2-c]benzopyran-2,5-dione, and 7H-pyrano[2,3-d]pyrimidin-7-one
References
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Transformation of Amines and N-Heteroarylformamidines into Esters of Substituted b-Amino-a,b-dehydro-a-amino Acids
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Synthesis of gamma-L-glutaminyl-[3,5-3H]4-hydroxybenzene and the study of reactions catalyzed by the tyrosinase of Agaricus bisporus.
TL;DR: Gamma-L-glutaminyl-3,4-dihydroxybenzene was synthesized in order to study the kinetics of its hydroxylation by tyrosinase purified from Agaricus bisporus and to explore its role in the induction of the dormant state in the spores of this species.
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Transformations of N‐heteroarylformamidines into derivatives of β‐heteroarylamino‐α,β‐dehydro‐α‐amino acids, β‐heteroarylamino‐α‐amino acids, and dipeptides
TL;DR: In this article, a general method for the preparation of β-heteroarylamino-α, β-dehydro-α-amino acids and dipeptides is described.
Journal Article
Intracellular Activation of γ-l-Glutaminyl-4-hydroxybenzene by Tyrosinase, a Mechanism for Selective Cytotoxicity against Melanocarcinoma
TL;DR: In tests of this hypothesis, the injection of γ-l-glutaminyl-4-hydroxybenzene with probenecid significantly inhibited the growth of human melanoma in athymic mice without apparent toxicity to the cells of the host that lack the enzyme.
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The synthesis of β‐heteroarylamino‐α,β‐dehydro‐α‐amino acid and β‐heteroarylamino‐α‐amino acid derivatives
TL;DR: The β-heteroarylaminomethyleneoxazolones as mentioned in this paper were obtained from heterogeneous formamidines and obtained by catalytic hydrogenation the compounds were converted into βhetero-arylamino substituted amides.