Journal ArticleDOI
The Baylis-HillmanBromides as Versatile Synthons: A Facile One-Pot Synthesisof Indolizine and Benzofused Indolizine Frameworks
TLDR
In this paper, a facile one-pot synthesis of indolizine, benzofused indoline and pyrrolo[1,2-a]quinoline derivatives from the Baylis-Hillman (B-H) bromides via an interesting strategy involving 1,5-cyclization of nitrogen ylides has been described.Abstract:
A facile one-pot synthesis of indolizine, benzofused indolizines {pyrrolo[1,2-a]quinoline and pyrrolo[1,2-a]isoquinoline} derivatives from the Baylis-Hillman (B-H) bromides, via an interesting strategy involving 1,5-cyclization of nitrogen ylides has been described.read more
Citations
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Journal ArticleDOI
Recent contributions from the Baylis-Hillman reaction to organic chemistry.
TL;DR: Acyclic activated alkenes/ alkynes and Asymmetric Baylis-Hillman Reaction: Earlier Developments 5495.
Journal ArticleDOI
Recent progress in synthesis and bioactivity studies of indolizines.
TL;DR: The present review describes the recent progress in synthetic approaches to construct indolizine framework (including partially or wholly reduced ring) and the design of such compounds with potential biological activity and emphasizes the importance of indolIZines in drug discovery.
Journal ArticleDOI
Cu(I)-catalyzed synthesis of imidazo[1,2-a]pyridines from aminopyridines and nitroolefins using air as the oxidant.
TL;DR: A copper-catalyzed method for the synthesis of imidazo[1,2-a]pyridine with aminopyridines and nitroolefins using air as oxidation agent in a one-pot procedure has been developed.
Journal ArticleDOI
Visible light mediated azomethine ylide formation—photoredox catalyzed [3+2] cycloadditions
TL;DR: The synthesis of highly functionalised N-heterocycles has been achieved by the visible light mediated photoredox conversion of tertiary amines to azomethine ylides and their further reaction with maleimide derivatives as dipolarophiles.
Journal ArticleDOI
Pyridine activation via copper(I)-catalyzed annulation toward indolizines.
TL;DR: The copper(I)-catalyzed regioselective [3 + 2] cyclization of pyridines toward alkenyldiazoacetates leading to functionalized indolizine derivatives is reported.
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