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Alan R. Katritzky
Researcher at University of Florida
Publications - 1988
Citations - 35516
Alan R. Katritzky is an academic researcher from University of Florida. The author has contributed to research in topics: Benzotriazole & Alkyl. The author has an hindex of 73, co-authored 1988 publications receiving 33831 citations. Previous affiliations of Alan R. Katritzky include University of North Texas & University of Akron.
Papers
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Journal ArticleDOI
The sulfonation of aromatic and heteroaromatic polycyclic compounds
Alan R. Katritzky,Myong Sang Kim,Dmytro Fedoseyenko,Khalid Widyan,M. Siskin,Manuel A. Francisco +5 more
TL;DR: In this paper, the relative reactivities of a series of polycyclic carbo-and heteroaromatic compounds to sulfonation by sulfur trioxide in nitrobenzene were measured and discussed.
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Lithium tetrafluoroborate-assisted reactions of N-(.alpha.-aminoalkyl)benzotriazoles with olefins and 1,3-dienes. New syntheses of 1,2,5,6-tetrahydropyridinium salts, 1,2,3,4-tetrahydroquinolines, and some related heterocyclic systems
Alan R. Katritzky,M. F. Gordeev +1 more
TL;DR: In this paper, the ionization of N-(α-aminoalkyl)benzotriazoles in tetrahydrofuran solution to generate reactive iminium intermediates, which can be trapped with electron-rich olefins and with 1,3-dienes.
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Design, synthesis, and biological activity of a novel series of 2,5-disubstituted furans/pyrroles as HIV-1 fusion inhibitors targeting gp41.
Shibo Jiang,Srinivasa R. Tala,Hong Lu,Peng Zou,Ilker Avan,Ilker Avan,Tarek S. Ibrahim,Tarek S. Ibrahim,Nader E. Abo-Dya,Nader E. Abo-Dya,Abdelmotaal Abdelmajeid,Abdelmotaal Abdelmajeid,Asim K. Debnath,Alan R. Katritzky,Alan R. Katritzky +14 more
TL;DR: A series of 2,5-disubstituted furans/pyrroles (5a-h) as HIV-1 entry inhibitors were designed and found to be effective in inhibiting HIV- 1 infection, with the best compounds being 5f and 5h, which exhibited significant inhibition on HIV-2(IIIB) infection at micromolar levels with low cytotoxicity.
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A C-13 nuclear magnetic resonance study of the pyrimidine synthesis by the reactions of 1,3-dicarbonyl compounds with amidines and ureas
TL;DR: In this paper, the detailed mechanistic pathways for the reactions of acetylacetone, methyl acetoacetate, and dimethyl malonate with a variety of amidines and ureas were elucidated.
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A Novel Transformation of Esters to Alkynes with 1-Substituted Benzotriazoles
TL;DR: In this article, the reaction of α-(benzotriazol-1-yl) 1-α-phenoxy hydrazones with methyllithium, n-butyllithium or phenyllithiam, alkynes were obtained, in which phenoxy groups were replaced by the lithium reagents.