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Alan R. Katritzky
Researcher at University of Florida
Publications - 1988
Citations - 35516
Alan R. Katritzky is an academic researcher from University of Florida. The author has contributed to research in topics: Benzotriazole & Alkyl. The author has an hindex of 73, co-authored 1988 publications receiving 33831 citations. Previous affiliations of Alan R. Katritzky include University of North Texas & University of Akron.
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A convenient synthesis of chiral 1,2,4-oxadiazoles from N-protected (α-aminoacyl)benzotriazoles
TL;DR: 1,2,4-Oxadiazoles derived from chiral α-amino acids were synthesized in 70–94% yields via a fast and easy procedure under mild conditions and were shown to be at least 97% enantiomerically pure by HPLC and NMR.
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N-triphenylphosphorylidene-1-(benzotriazol-1-yl)methylamine, a novel synthon equivalent to +CH2NH2: The preparation of primary amines
TL;DR: In this article, primary amines are readily prepared by reaction of the title compound with organolithiums or Grignard reagents, and they can be used to synthesize primary amine derivatives.
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Synthesis and physicochemical properties of thiadiazolo[3,2-a]pyrimidinesulfonamides and thiadiazolo[3,2-a]triazinesulfonamides as candidates for topically effective carbonic anhydrase inhibitors.
TL;DR: A number of compounds synthesized from 5-amino-1,3,4-thiadiazole-2-sulfonamide exhibited lower sulfonamide pKa and higher water solubility than those of acetazolamide and methazlamide, and one, 12, brought about a small reduction in IOP in the normal rabbit eye.
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Conformational analysis of saturated heterocycles. XX. Stereochemistry of base-catalyzed hydrogen-deuterium exchange of methylene protons .alpha. to a sulfinyl group
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Efficient Syntheses of Imidazolo[1,2-a]pyridines and -[2,1-a]isoquinolines
TL;DR: 2-Aminopyridines 1a-c and 1-aminoisoquinoline with 1-chloromethylbenzotriazole give 2-amino-1-[alpha-benzol-1-ylmethyl]pyridinium chlorides + chloride 12, respectively, which enable imidazolo[2, 1-a]isoquinolines 13a,b in good yields.